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TECHNIC SUPORTER
BEIKING UNIVERSITY
JINAN UNIVERSITY
XIAMEN UNIVISITY
CHINA AGRICULTURAL UNIVERSITY
CHINESE ACADEMY OF SCIENCES
SHANGHAI INSTITUTE OF MATERIA MEDICA
LIAONING UNIVERSITY
SHENYANG PHARMACEUTICAL UNIVERSITY
INTERMEDIATES


ACYCLOVIR
2-oxa-1,4-butanedil diacetate
ADENOSINE
6-chloropurine

ALLOPURINOL
3-mopholine-2-cyanocrylamide
5-amino-4-pyrazole carboxamide hemisalfate
ethoxymethylene cyanoacetic acid ethyl ester

ALOSETRON
2,3,4,5-tetrahydro-5-methyl-1h-pyrido[4,3-b]indol-1-one

ALPRAZOLAM
2-chloroacetylamine-5-chlorobenzophenone
2-amino-5-chlorobenzophenone

AMANTADINE
adamantane
1-bromo adamantane
adamantylamine

AMBROXOL
trans-4-amino cyclohexyphenol
2-amino-3,5-dibromo benzaldehyde

AMILORIDE
3-amino-5,6-dichloropyrazine2-methyl formate
3,5-diamino-6-chloropyrazine-2-methyl formate

AMIODARONE
2-butyl-3-(p-hydroxybenzoyl)benzofuran
2-butyl-3-(3',5,5-diido-4-hydroxybenzoyl) benzofuran

AMITRIPTYLINE
3-dimethylaminopropyl Chloride Hcl min98.0%
Dibenzosuberone min97.0%


ATENOLOL
4-aminophenyl acetic acid
4-hydroxyphenyl acetamide

ATORVASTATIN
(r)-4-cyano-3-hydroxybutyric acid ethyl ester
(4r-cis)-1,1-dimethylethyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxane-4-acetate
(4r-cis)-1,1-dimethylethyl-6-aminoethyl-2,2-dimethyl-1,3-dioxane-4-acetate
4-fluoro-alpha-[2-methyl-1-oxopropyl]-gama-oxo-n,beta-diphenyl benzene butaneamide
(4r-cis)-1,1-dimethylethyl-6-[2-(4-fluorophenyl)-5-(1-methylethyl)-3-phenyl-4-[(phenylamino) carbonyl]-1h-pyrrol-1-yl]ethyl]-2,2-dimethyl-1,3-dioxane-4-acetate

AZATHIOPRINUM
5-chloro-1-methyl imidazole
5-chloro-1-methyl-4-nitroimidazole

BAMBUTEROL
3,5-dihydroxy benzoic acid
3,5-dihydroxy acetophenone
3,5-diphenoxy acetophenone

BENAZEPRIL
4-hydroxyphenethylamine
tert-butyl-(s)-(3-amino-2-oxo-2,3,4,5-tetrahydro benzo[b]azepin-1-yl)acetate

BRODIMOPRIM
4-bromo-3,5-dihydroxybenzoic acid
4-bromo-3,5-dimethoxybenzoic acid
4-bromo-3,5-dimethoxy benzoyl chloride
4-bromo-3,5-dimethylbenzaldehyde

BROMHEXINE
2-amino-3,5-dibromotoluene
2-diacetylamino-3,5-dibromobenzyl bromide
n-methyl-n-cyclohexyl-2-amino-3,5-dibromophenylmethylamine

BUFLOMEDIL
1,3,5-trimethoxybenzene
4-chlorobutyryl chloride
1-(4-chlorobutyryl)-2,4,6-trimethoxybenzene

BUMETANIDE
4-chloro-3,5-dinitrobenzoic acid
4-phenoxy-3,5-dinitrobenzoic acid
5-nitro-4-phenoxy-3-aminosulfonyl benzoic acid
5-amino-4-phenoxy-3-aminosulfonyl benzoic acid

BUTENAFINE
4-(tert-butyl)benzyl chloride
4-(tert-butyl)benzyl bromide
n-methyl-1-naphthalenemethylamine hcl

CANDESARTAN
2-cyano-4ĄŻ-bromomethylbiphenyl

CAPTOPRIL
d-3-acetylthio-2-methyl propionyl-l-proline

CARBAMAZEPINE
iminodibenzyl
chlorocabonyl liminostilben

CARVEDIOL
4-hydroxycarbazole
1,2,3,4-terahydro-4-oxocarbazole
2-(2-methoxyphenoxy)ethylamine hcl

CEFOTAXIME
s-(2-benzothiazole yl)-2-(2-aminothiazol-4-yl)-(z)-2-methoxyimino thioacetate
2-methoxyimino-2-(2-aminothiazole-4-yl)-acetic acid anhydrous

CEFOTIAM
d-(-)-a-(4-ethyl-2,3-dioxo piperzinyl) carboxyamide-4-hydroxyphenyl acetic acid
2-amino-4-thiazolyl-acetic acid

CHLORDIAZEPOXIDE
2-amino-5-chlorobenzophenone min98.5%


CHLORPROTHIXENE
2-chloro-9h-ph-thioxanthen-9-one-(2-chlorothioxathone)
2-chloro-9-(3-dimethylaminopropyl)-ph-thioxanthe-9-ol

CHLORTHALIDONE
2-(3-amino-4-chlorobenzoyl) benzoic acid

Cimetidine
cyanoiminodithio carbonic acid dimethyl ester
Cysteamine HCL
S-Methyl


CLOFIBRATE
clofibric acid

CLONAZEPAM
2-amino-5-nitro-2'-chlorobenzophenone

CLOPIDOGREL
2-thiophene ethanol
2-thiophene ethylamine
r,s-2-chloro-(alpha bromo)phenylacetic acid
(dl)-methyl-alpha-(2-thienylethamino)(2-chlorophenyl)acetate hcl

CYCLANDELATE,PEMOLINE
DL-Mandelic acid


CYCLOPHOSPHAMIDE
bis-(chloroethyl)amine hcl

CYPROHEPTADINE
Dibenzosuberonone min97.0%


CYPROTERONE ACETATE
1,6-didehydro-17a-hydroxy progesterone
1,6-didehydro-17a-acetoxy progesterone
1,2-a-methylene-6-didehydro-17a-acetoxy progesterone
1-chloromethyl-6-chloro-6-dehydro-17a-acetoxy progesterone

DACARBAZINE
4-formamido-5-aminoimidazole hcl
5-aminoimidazole-4-foramido hcl

Diazepam
2-methylamino-5-chlorobenzophenone min99.0%
3-benyl-5-chlorobenzoixoxazole mp112.0-114.0


DICLAZURIL
2,6-dichloro-alpha-(4-chlorophenyl)-4-nitrophenzyl cyanide
4-amino-2,6-dichloro-alpha-(4-chlorophenyl)phenzyl cyanide

Dihydralazine sulfate
Phthalhydrazide(1,4-Dionephthalaxine)


DOMPERIDONE
1-benzyl-3-methoxycarbonyl-4-piperidone
2-b-(chloropropyl)-1,3-dihydro-2h-benzimidzole-2-one
1-(4-piperidinyl)-1,3-dihydroxy-2h-5-chloro benzimidazolone

DOXAZOSIN
2-amino-4,5-dimethoxybenzoic acid
2-chloro-4-amino-6,7-dimethoxyquinazoline

DOXEPIN
phthalide
11-dihydrodibenz[b,c]oxcpin-11-one
11-(3-dimethylaminopropyl-6,11-dihydrodibenz[b,c]oxcpin-11-ol

ENALAPRIL
n-[1-(s)-ethoxycarbonyl-3-phenylpropyl]-l-alanine

ESMOLOL
3-[4-[2-hydroxy-3-[(1-methylethyl)amino] propoxy]phenyl]acrylate hcl

FAMCICLOVIR
2-amino-6-hydroxypurine
6-chloropurine
2,6-dichloropurine
2-amino-6-chloropurine
9-(4-acetoxy-3-acetoxymethylbut-1-yl)-2-amino-6-chloropurine

Famotidine
1,3-dichoro acetone
guanyl thiourea
N-sulfamyl-3-chloropropionamidine hydrochloride
Omeprazole(Omeprazole Sodium)
S-(2-guanidino-4-thiazol methyl)Isothiourea Dihydrochloride
sulfamide


FELODIPINE
2,3-dichlorobenzaldehyde

FENOFIBRATE 4-chloro-4'-hydroxybenzophenone
2-[4-(p-chlorobenzoyl) phenoxy]-2'-methyl-propionue acid

FINASTERIDE
androst-3-one-4-ene-17b-carboxylic acid
androst-4-aza-3-one-17b-butyl carboxamide
3-oxo-4-aza-5a-androstane-17b-carboxylic acid

FIPRONIL
2,6-dichloro-4-trifluoromethyl aniline

FLECAINIDE
2,5-bis-(2,2,2-trifluoroethoxy)benzoic acid

FLUCONAZOLE
2,4-difluoro-a-(1h-1,2,4-triazol-1yl) acetophenone

FLUNARIZINE
n-mono-[4,4'-fluorobenzyl] methyl piperazine

FLUOROURACIL
2-mercapto-4-hydroxy-5-fluoropyrimidine

FLUOXETINE
3-methylamino-1-phenyl-propanol
3-hydroxy-n-methyl-3-phenyl propylamine
Alpha-[2-(methylamino)-ethyl]benzyl alcohol


FLURAEPAM
2-amino-5-chloro-2'-fluorobenzophenone

FLURAZOPAN
2-amino-5-chloro-2ĄŻ-fluorobenzophenone
7-chloro-5-(2-fluorophenyl)1,3-dihydro-1,4-benzodiazepine-2-one

FLUROBENDAZOLE
4-chloro-4ĄŻ-fluoro-3-nitrobenzophenone

FLUTAMIDE
3-trifluoromethyl-4-nitro aniline

FORMOTEROL
3-nitro-4-hydroxyacetophenone

FUROSEMIDE
2,4-dichloro-5-sulfamide benzoic acid
2,4-dichloro-5-aminosulfomylbenzoic acid
2-amino-4-chloro-5-aminosulfomyl benzoic acid

GABAPENTINE
1,1-cyclohexane diacetic acid monoamide
1-cyanocyclohexane acetonitrele
1-cyanocyclohezne acetic acid ester
1,1-cyclohexane diacetic anhydride
3,3-pentamethylene glutarimide
4,4-pentamethylene-2-pyrrolidinone

GATIFLOXACINE
2,4,5-trifluoro-3-methoxybenzoic acid
1-cyclopropyl-6,7-difluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinoline carboxylic acid ethyl ester

GEMFIBROZIL
2,5-dimethyl phenol
isobutyl-5-chloro-2,2-dimethylvalerate

GLIBENCAMIDE
5-chloro-2-methoxy
4-(2-aminoethyl)benzene sulfonamide
4-[2-(5-chloro-2-methoxy benzamide)ethyl]benzene sulfonamide

GLICLAZIDE
n-amino-3-azabciclo(3,3,0) octane hcl

GLIMEPIRIDE
3-ethyl-4-methyl-2-oxo-pyrroline
trans-4-methyl cyclohexylamine

GLIQUIDONE
4,4-dimethyl-7-methoxyisochroman-1,3-dione
n-[2-(4-sulfonamidylphenyl)ethyl]-4,4-dimethyl-7-methoxy-1,2,3,4- tetrahydroisoquinoline-1,3-dione

GRANISETRON
1-methyl-1h-indazole-3-carboxychloride

HALOPERIDOL
4-(4-chlorophenyl)-4-hydoxypiperidine

IMIQUIMOD
3-amino-2-chloro-4-[(2-methylpropyl)amino]quinoline

IRBESARTAN
2-cyano-4ĄŻ-bromomethylbiphenyl
2-butyl-1,3-diazapiro[4,4]non-1-en-4-one hcl
2-(1h-1-triphenyl-tetrazol-5-yl)-4ĄŻ-bromomethyl diphenylene
1-amino-1-cyclopentane carboxamide

IRINOTECAN
campthotecin
7-ethylcampthotecin
7-ethyl-10hydroxycampthotecin

ITRACONAZOLE
cis-[2-(2,4-dichlorophenyl)-2-(1h-1,2,4-triazole-1-ylmethyl)-1,3-dioxolan-4-yl]- -methyl methanesulfonate
2,4-dihydro-4-[[4-(4-hydroxyphenyl)-1-piperazinyl]-phenyl]-2-(1-methylpropyl)- -3h-1,2,4-triazole-3-one

KETOCOANZOLE
1-acetyl-4-(4-hydroxyphenyl) piperazine
[is-2-(2,4-dichlorophenyl)-2-1h-imidazole-1-yl-methyl-1,3-dixoan-4-yl] methyl -phenylmethane sulfonate

LANSOPRAZOLE
2,2,2-trifluoroethanol
2-hydroxymethyl-3-methyl-4-(2,2,2-trifluoroethoxy)pyridine
2-chloromethyl-3-methyl-4-(2,2,2-trifluoroethoxy)pyridine


LEFLUNOMIDE
5-methylisooxazole-4-benzoic acid

LEVOFLOXACIN
s-(+)-2-amino propanol

LINEZOLID
3,4-difluoro nitro benzene

LISINOPRIL
ethoxy carbonyl phenyl propyl-n-trifluoro acetyl-l-lysine

LOPERAMIDE
4-chlorophenyl-4-hydroxy piperidine
3,3-diphenyl-2-furlidine amino bromide

LORATDINE
2-cyano-3-methylpyridine
n-methyl-4-chloro-piperdine hcl
5-amino-4,6-dichloro-2-methyl pyrimidine
3-[2-(3-chlorophenyl)ethyl]-2-pyridine carbonitrile
3-[2-(3-chlorophenyl)ethyl]-2-pyridine carboxchloride
8-chloro-6,11-dihydro-5h-benzo-(5,6)cyclohepta(1,2-pyridine-11-one)

LOSARTAN
2-cyano-4ĄŻ-methylbiphenyl
2-cyano-4ĄŻ-bromomethylbiphenyl

MELOXICAM
2-amino-5-methylthiazole
2-methyl-4-hydroxy-2h-1,2-benzothiazine-3-carboxylic acid ethyl ester-1,1-dioxide

METHYLDOPA
3-hydroxy-4-methoxybenzaldehyde
3,4-methylenedioxyphenyl-2-propanone

METOPROLOL
4-(2-methoxyethyl)phenol

MIDAZOLAM
2-amino-5-chloro-2ĄŻ-fluorobenzophenone
2-aminomethyl-7-chloro-2,3-dihydro-5-(2-fluorophenyl)-1h-1,4-benzodiazepine dimaleate
7-chloro-1,3-dihydro-5-(2-fluorophenyl)-2-nitromethylene-2h-1,4-benzodiazepine
8-chloro-3a,4-dihydro-6-(2-fluorophenyl)-1-methyl-3h-imidaz[1,5a][1,4]benzodiazepine

MODAFINIL
diphenylmethanol
diphenylmethyl thioacetic acid
ethyl diphenylmethyl thioacetate

MOXIFLOXACIN
2,3-pyridinedicarboxylic anhydride cas: 699-98-9

MOXONIDINE
5-amino-4,6-dichloro-2-methylpyrimidine

NATEGLINIDE
trans-4-(1-methylethyl)cyclohexane carboxylic acid

NEBIVOLO
5-fluoro-2-hydroxy acetophenone

NELFINAVIR
3-acetoxy-2-methylbenzoic acid

Nitrazepam
2-amino-5-nitrobenzophenone min99.0%


NIZATIDINE
dimethyl aminoacetonitrile
dimethyl aminothio acetmide
2-dimethylaminomethyl-4-chloromethyl-4-hydroxyl thiazoline
2-dimethylaminomethyl-4-chloromethylthiazole hcl
2-(n,n-dimethylaminomethyl)-4-carbethoxy thiazole
s-(2-dimethylaminomethyl)-4-thiazolemethyl isothioure dihcl
2-(dimethylaminomethyl)4-thiazolemethanol
n-(2-thioethyl)-nĄŻ-methyl-2-nitro-1ĄŻ,1-ethendiamine
n-(2-chloroethyl)-nĄŻ-methyl-2-nitro-1ĄŻ,1-ethendiamine

OMEPRAZOLE
2-chloromethyl-3,5-dimethyl-4-methoxy pyridine hcl
3,5-dimethyl-4-methoxy pyridine-2-chloro methyl hcl
2,3,5-Trimethyl pyridine
2-Mercapto-5-methoxybenzimidazole
4-methoxy-3,5-dimethyl-2-hydromethyl pyridine


ONDANSETRONE
1,2,3,9-trtrahydro-9-methyl-4h-carbazol-4-one
3-[(dimethylamino)methyl]-1,2,3,9-tetrahydro-9-methyl-4h-carbazole-4-one

OXYBUTYNIN
cyclohexylmandelic acid methyl ester

PANTOPRAZOLE
2-chloromethyl-3,4-dimethoxy pyridine hcl
3-methoxy-2-methyl-4-(1h)-pyridone
4-chloro-3-methoxy-2-methyl pyridine-n-oxide
5-difluormethoxy-2-mercapto-1h-benzimidazole

PAROXETINE
trans-4-(4-fluorophenyl)-3-hydroxymethyl piperidine
4r-(4ĄŻ-fluorophenyl)-3s-[(3ĄŻ,4ĄŻ-methylenedioxyphenoxyl)methyl]-n-methylpiperidine

PENCICLOVIR
2-amino-6-chloropurine

PERPHENAZINE
n-(2-hydroxyethyl) piperazine

PIROXICAM
2-methyl-4-hydroxy-2h-1,2-benzothiazine-3-carboxylic acid ethyl ester-1,1-dioxide

PRAZOSIN
4-amino-2-chloro-6,7-dimethoxyquinazoline

QUETIAPINE
2-(2-chloroethoxy)ethanol
dibenzo[b,f][1,4]thiazepine-11(oh)-one

RALOXIFENE
4-(2-piperidinoethoxy)benzoic acid
6-methoxy-2-(4-methoxyphenyl)benzothiophene

RANITIDINE
1-methoxy-1-methylamino-2-nitroethylene
1,1-dimethylthio-2-nitroethylene
1-methylamino-1-methylthio-2-nitroethylene
Cysteamine HCL


RIFAMPICIN
1-amino-4-methylpiperazine

RIMANTADINE
1-bromo adamantane
1-adamantyl methyl ketone
1-adamantane carboxulic acid

SERTRALINE
4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-naphthalone
4-(3,4-dichlorophenyl)-1-tetralone

SIBUTRAMINE
1-(4-chlorophenyl)cyclobutanecarbonitril

SILDENAFIL
4-amino-1-methyl-3-n-propylpyrazole-5-carboxamide
5-(2-ethoxyphenyl)-1methyl-3-propyl-6,7-dihydro-1h-pyrazolo pyrimidin-7-one

SOTALOL
4-(chloroacetyl)phenylmethane sulfonamide
4-(isopropylamino)phenylmethane sulfonamide

STARVUDINE
3ĄŻ,5-dimethane sulfonyl thymidine
2-dexoy-3,5-epoxythymine

SULPIRIDE
1-ethyl-2-aminmethylene pyrrolidine
2-methoxy-5-sulfamoyl benzoic acid

SUMATRIPAN
4-hydrazino-n-methyl-benzene methane sulfonamide hcl
4(dimethyl amino)butyraldehyde dimethyl acetal

T.M.P
3,4,5-trimethoxy-2-methoxymethyl cynnamonitrile

TAZOBACTAM
benzhydryl-6,6-dibromopenicillanate-1-oxide

TEGASEROD
5-methoxy-3-indole carboxaldehyde

TELMISARTAN
2-cyano-4ĄŻ-bromomethylbiphenyl
1H-benzimidazole-5-carboxylic acid, 7-methyl-2-propyl CAS 152628-03-0

TERAZOSINE
4-amino-2-chloro-6,7-dimethxoyquinazoline
2-amino-4,5-dimethoxybenzoic acid

TERBINAFINE
3,3ĄŻ-dimethyl-1-butynene
trans-1,3-dichloropropylene
methyl naphthalene-1-yl-methylamine

THIOCTIC ACID
6,8- dichloro ethyl caprylate

THIORIDAZINE
2-thomethyl phenothiaize
bata-ethylchloride-n-methyl piperidine hcl

TIAPRIDE
2-methoxy-5-methylsulfonyl benzoic acid

TIBOLONE
7a-methyl-3,3-dimethoxy-5(10)-estrene-17-one

TIMOLOL
3,4-dichloro-1,2,5-thiadiazole
3-morpholine-4-chloro-1,2,5-thiadiazole
s-(-)-tert-butylamine-1,2-propylene glycol

TOPOTECAN
iodobenzene camptothecinum 10-hydroxycamptothecinum

TORASEMIDE
4-[(3-methylphenyl)amino]-3-pyridinesulfonamide

TORSEMIDE
4-(3-methylphenyl)aminopyridine-3-sulfonamide

TOSUFLOXACIN
ethyl-(2,6-dichloro-5-fluoronicotinoyl)acetate

TRAPIDIL
3-amino-1h-1,2,4-triazole

TRIAMTERENE
2,4,6-triaminopyrimidine
2,4,6-triamino-5-nitropyrimidine

TRIAZOLAM
2-amino-5-chloro-2'-chloro benzopheone

TRIMEBUTINE
3,4,5-trimethoxy benzoic acid

TROVAFLOXACIN
3-hydroxy acetophenone
3-amino acetophenone

VALACICLOVIR
2-amino-6-chloropurine

VALSARTAN
2-(1h-1-triphenyl-tetrazol-5-yl)-4ĄŻ-bromomethyl diphenylene

VENAFAXINE
1-[cyano-(4-methoxyphenyl)]cyclohexanol
1-[2-amino-1-(4-methoxyphenyl)ethyl]cyclohexanol
n,n-dimethyl-2-(1-hydroxy cyclohexyl)-2-(4-methoxy) acetamide

VITAMIN D2
3,5-dinitrobenzoic acid
3,5-dinitrobenzoyl chloride

VITAMIN H
cis-1,3-dibenzylimidazole-2-one-4,5-dicarboxylic acid

WARFARIN
4-hydroxycoumarin

ZALEPLON
3-amino-1h-pyrazole-4-carbonitrile

ZIPRASIDONE
1,2-benziothiazole.3-(1-piperazinyl), hcl CAS 87691-88-1
2H-indole-2-one,5-chloroethyl-6-chloro-1,3-dihydro CAS 118289-55-7

ZOLPIDEM
2-(4-methylphenyl)-6-methylimidazole pyridine
2-(4-methylphenyl)-6-methylimidazole pyridine-3-acetonitrile

ZOPICLONE
2,3-pyrazine dicarboxylic anhydride
2-amino-5-chloropyridine
6-(5-chloro-2-piperidinyl)-6,7-dihydro-7-hydroxy-5h-pyrrolo[3,4-b]pyrazine-5-one

 

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